GRIECO, PAOLO
GRIECO, PAOLO
DIPARTIMENTO DI FARMACIA
Cyclic peptides acting as urotensin-II antagonists.
2005 Novellino, Ettore; Grieco, Paolo; Rovero, P.
Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives
1996 Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa
D-Amino Acid Scan of g-Melanocyte-Stimulating hormone:importance of the Trp8
2000 Grieco, Paolo; Balse, P. M.; Weinberg, D.; Macneil, T.
" Molecular Modelingof the Urotensin-II receptor Complex"
2004 Grieco, Paolo; Lavecchia, A.; Campiglia, P.; Lama, T.; Rovero, P.; Carotenuto, Alfonso; Patacchini, R.; Maggi, C. A.; Novellino, Ettore
A structure – activity relationship study on position –2 of the Gas C-terminal peptide able to inhibit Gs activation by A2A adenosine receptor.
2003 Grieco, Paolo; Albrizio, Stefania; D’Ursi, A. M.; Giusti, L.; Mazzoni, M. R.; Novellino, E.; Rovero, P.
Cross-talk between fmlp and αvβ5 receptors triggered by urokinase receptor-derived SRSRY peptide
2005 Gargiulo, L.; Longanesi, Cattani; I., Bifulco; K., Franco; P., Raiola; R., Romano; A., Campiglia; Grieco, Paolo; P., Peluso; G., Stoppelli; M. P., Carriero; M., V.
Conformational analysis of the new temporin analogues: Gln3TA and Pro3TL
2008 M. R., Saviello; A., Cavalli; S., Malfi; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; M. L., Mangoni; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso
Design, Synthesis, and Conformational Analysis of Melanotropin Analogues of MTII and SHU9119
2013 Grieco, Paolo; Minying, Cai; Yousif, ALI MUNAIM; Carotenuto, Alfonso; Limatola, Antonio; Brancaccio, Diego; Novellino, Ettore; Victor J., Hruby
Unraveling the active conformation of urotensin II
2004 Carotenuto, Alfonso; Grieco, Paolo; Campiglia, Pietro; Novellino, Ettore; Ettore, Rovero; Paolo,
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan.
1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands.
2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Further Evidence that Melanocortins Prevent Myocardial Reperfusion Injury by Activating MC3 Receptors: Irrelevance of the C-terminal Arg-Phe sequenze
2003 Mioni, C; Giuliani, D; Cainazzo, M. M; Leone, S; Iannone, C; Bazzani, C; Grieco, Paolo; P, Novellino; E, Tomasi; A, Bertolini; A, Guarini
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Synthesis and Pharmacological Evaluation of Analogs of Indole-Based Cannabimimetic Agents.
2010 Mazzoni, O; Diurno, MARIA VITTORIA; di Bosco, Am; Novellino, Ettore; Grieco, Paolo; Esposito, G; Bertamino, A; Calignano, Antonio; Russo, Roberto
Structure-Activity Relationships of Novel Cyclic alpha-MSH/gamma-MSH Hybrid Analogues which Lead to Potent and Selective Ligands for the Human MC3R and Human MC5R
2003 Balse, Srinivasan; P., M.; Grieco, Paolo; P, Cai; M, Trivedi; D, Hruby; V., J.
Extensive Structure-Activity Studies of Lactam Derivatives of MT-II and SHU9119: Their activity and Selectivity at Human Melanocortin Receptors 3,4 and, 5.
2003 Grieco, Paolo; P, Balsesrinivasan; P, Han; G, Weinberg; D, Macnail; T, ; VAN DER, Ploeg; L. H. T, Hruby; V., J.
Development of Cyclic Peptide Inhibitors of GRK2
2013 Carotenuto, Alfonso; Limatola, Antonio; Cipolletta, Ersilia; Sala, Marina; Vernieri, Ermelinda; GOMEZ MONTERREY, ISABEL MARIA; Bertamino, Alessia; Musella, Simona; Grieco, Paolo; Novellino, Ettore; Iaccarino, Guido; Campiglia, Pietro
NMR analysis of synthetic peptides agonist to PTPRJ, a receptor-type protein tyrosine phosphatase with tumor suppressor activity
2011 Brancaccio, Diego; Carotenuto, Alfonso; Grieco, Paolo; Campiglia, P; Trapasso, F; Novellino, Ettore
Melanocortin type 3 receptor null mice are refractory to the inhibitory actions of a selective receptor agonist in experimental acute inflammation
2006 Getting, J. S.; Lam, C. W.; Chen, A. S.; Grieco, Paolo; Perretti, M.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Cyclic peptides acting as urotensin-II antagonists. | 6.1 Brevetto | 2005 | Novellino, Ettore; Grieco, Paolo; Rovero, P. | |
| Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives | 1.1 Articolo in rivista | 1996 | Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa | |
| D-Amino Acid Scan of g-Melanocyte-Stimulating hormone:importance of the Trp8 | 1.1 Articolo in rivista | 2000 | Grieco, Paolo; Balse, P. M.; Weinberg, D.; Macneil, T. | |
| " Molecular Modelingof the Urotensin-II receptor Complex" | 4.1 Articoli in Atti di convegno | 2004 | Grieco, Paolo; Lavecchia, A.; Campiglia, P.; Lama, T.; Rovero, P.; Carotenuto, Alfonso; Patacchini, R.; Maggi, C. A.; Novellino, Ettore | |
| A structure – activity relationship study on position –2 of the Gas C-terminal peptide able to inhibit Gs activation by A2A adenosine receptor. | 1.1 Articolo in rivista | 2003 | Grieco, Paolo; Albrizio, Stefania; D’Ursi, A. M.; Giusti, L.; Mazzoni, M. R.; Novellino, E.; Rovero, P. | |
| Cross-talk between fmlp and αvβ5 receptors triggered by urokinase receptor-derived SRSRY peptide | 1.1 Articolo in rivista | 2005 | Gargiulo, L.; Longanesi, Cattani; I., Bifulco; K., Franco; P., Raiola; R., Romano; A., Campiglia; Grieco, Paolo; P., Peluso; G., Stoppelli; M. P., Carriero; M., V. | |
| Conformational analysis of the new temporin analogues: Gln3TA and Pro3TL | 4.1 Articoli in Atti di convegno | 2008 | M. R., Saviello; A., Cavalli; S., Malfi; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; M. L., Mangoni; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso | |
| Design, Synthesis, and Conformational Analysis of Melanotropin Analogues of MTII and SHU9119 | 1.5 Abstract in rivista | 2013 | Grieco, Paolo; Minying, Cai; Yousif, ALI MUNAIM; Carotenuto, Alfonso; Limatola, Antonio; Brancaccio, Diego; Novellino, Ettore; Victor J., Hruby | |
| Unraveling the active conformation of urotensin II | 1.1 Articolo in rivista | 2004 | Carotenuto, Alfonso; Grieco, Paolo; Campiglia, Pietro; Novellino, Ettore; Ettore, Rovero; Paolo, | |
| Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania | |
| Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. | 1.1 Articolo in rivista | 2000 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R. | |
| Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G. | |
| Further Evidence that Melanocortins Prevent Myocardial Reperfusion Injury by Activating MC3 Receptors: Irrelevance of the C-terminal Arg-Phe sequenze | 1.1 Articolo in rivista | 2003 | Mioni, C; Giuliani, D; Cainazzo, M. M; Leone, S; Iannone, C; Bazzani, C; Grieco, Paolo; P, Novellino; E, Tomasi; A, Bertolini; A, Guarini | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Synthesis and Pharmacological Evaluation of Analogs of Indole-Based Cannabimimetic Agents. | 1.1 Articolo in rivista | 2010 | Mazzoni, O; Diurno, MARIA VITTORIA; di Bosco, Am; Novellino, Ettore; Grieco, Paolo; Esposito, G; Bertamino, A; Calignano, Antonio; Russo, Roberto | |
| Structure-Activity Relationships of Novel Cyclic alpha-MSH/gamma-MSH Hybrid Analogues which Lead to Potent and Selective Ligands for the Human MC3R and Human MC5R | 1.1 Articolo in rivista | 2003 | Balse, Srinivasan; P., M.; Grieco, Paolo; P, Cai; M, Trivedi; D, Hruby; V., J. | |
| Extensive Structure-Activity Studies of Lactam Derivatives of MT-II and SHU9119: Their activity and Selectivity at Human Melanocortin Receptors 3,4 and, 5. | 1.1 Articolo in rivista | 2003 | Grieco, Paolo; P, Balsesrinivasan; P, Han; G, Weinberg; D, Macnail; T, ; VAN DER, Ploeg; L. H. T, Hruby; V., J. | |
| Development of Cyclic Peptide Inhibitors of GRK2 | 1.5 Abstract in rivista | 2013 | Carotenuto, Alfonso; Limatola, Antonio; Cipolletta, Ersilia; Sala, Marina; Vernieri, Ermelinda; GOMEZ MONTERREY, ISABEL MARIA; Bertamino, Alessia; Musella, Simona; Grieco, Paolo; Novellino, Ettore; Iaccarino, Guido; Campiglia, Pietro | |
| NMR analysis of synthetic peptides agonist to PTPRJ, a receptor-type protein tyrosine phosphatase with tumor suppressor activity | 1.5 Abstract in rivista | 2011 | Brancaccio, Diego; Carotenuto, Alfonso; Grieco, Paolo; Campiglia, P; Trapasso, F; Novellino, Ettore | |
| Melanocortin type 3 receptor null mice are refractory to the inhibitory actions of a selective receptor agonist in experimental acute inflammation | 1.1 Articolo in rivista | 2006 | Getting, J. S.; Lam, C. W.; Chen, A. S.; Grieco, Paolo; Perretti, M. |