SANTAGADA, VINCENZO
SANTAGADA, VINCENZO
DIPARTIMENTO DI FARMACIA
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV
2001 Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones.
2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6
2015 Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
Synthesis and Biological Effects of Hydrogen Sulfide (H2S): Development of H2S-Releasing Drugs as Pharmaceuticals
2010 Caliendo, Giuseppe; Cirino, Giuseppe; Santagada, Vincenzo; Wallace, J. L.
Synthesis of benzamide derivatives and their evaluation as antiprion agents
2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346)
2010 Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe
Synthesis and neurokinin antagonist activity of 2-benzylidene- and 2- benzyl-3-benzylamino quinuclidines
1993 Caliendo, Giuseppe; Greco, Giovanni; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Turbanti, L.; Renzetti, A. R.; Benedetti, E.; Pedone, C.; Santini, A.
Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives
1996 Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa
Na+/Ca2+ exchanger in Na+ efflux-Ca2+ influx mode of operation exerts a neuroprotective role in cellular models of in vitro anoxia and in vivo cerebral ischemia.
2002 Tortiglione, A.; Pignataro, Giuseppe; Minale, M.; Secondo, Agnese; Scorziello, Antonella; DI RENZO, GIANFRANCO MARIA LUIGI; Amoroso, S.; Caliendo, Giuseppe; Santagada, Vincenzo; Annunziato, Lucio
S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids.
2001 Alves, L. C.; Melo, R. L.; Sanderson, S. J.; Mottram, J. C.; Coombs, G. H.; Caliendo, Giuseppe; Santagada, V.; Juliano, L.; Juliano, M. A.
Protease activated receptor-2 modulates myocardial ischemia reperfusion injury in the rat heart.
2000 Napoli, C; Cicala, Carla; Wallace, J; DE NIGRIS, F; Santagada, V; Caliendo, G; Franconi, F; Ignarro, L; Cirino, Giuseppe
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei
2000 Balboni, G.; Salvadori, S.; Guerrini, R.; Bianchi, C.; Santagada, V.; Caliendo, Giuseppe; Bryant, S. D.; Lazarus, L. H.
5-amino-2-hydroxybenzoic acid 4-(5-thioxo-5H-[1,2]dithiol-3yl)-phenyl ester (ATB-429), a hydrogen sulfide-releasing derivative of mesalamine, exerts antinociceptive effects in a model of postinflammatory hypersensitivity
2006 Distrutti, E; Sediari, L; Mencarelli, A; Renga, B; Orlandi, S; Russo, G; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, G; Wallace, Jl; Fiorucci, S.
Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study
1997 Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A.
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
| Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV | 1.1 Articolo in rivista | 2001 | Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S. | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe | |
| Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 | 1.1 Articolo in rivista | 2015 | Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano | |
| Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists | 1.1 Articolo in rivista | 2001 | Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa, | |
| Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
| Synthesis and Biological Effects of Hydrogen Sulfide (H2S): Development of H2S-Releasing Drugs as Pharmaceuticals | 1.1 Articolo in rivista | 2010 | Caliendo, Giuseppe; Cirino, Giuseppe; Santagada, Vincenzo; Wallace, J. L. | |
| Synthesis of benzamide derivatives and their evaluation as antiprion agents | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe | |
| Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346) | 1.1 Articolo in rivista | 2010 | Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe | |
| Synthesis and neurokinin antagonist activity of 2-benzylidene- and 2- benzyl-3-benzylamino quinuclidines | 1.1 Articolo in rivista | 1993 | Caliendo, Giuseppe; Greco, Giovanni; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Turbanti, L.; Renzetti, A. R.; Benedetti, E.; Pedone, C.; Santini, A. | |
| Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives | 1.1 Articolo in rivista | 1996 | Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa | |
| Na+/Ca2+ exchanger in Na+ efflux-Ca2+ influx mode of operation exerts a neuroprotective role in cellular models of in vitro anoxia and in vivo cerebral ischemia. | 1.1 Articolo in rivista | 2002 | Tortiglione, A.; Pignataro, Giuseppe; Minale, M.; Secondo, Agnese; Scorziello, Antonella; DI RENZO, GIANFRANCO MARIA LUIGI; Amoroso, S.; Caliendo, Giuseppe; Santagada, Vincenzo; Annunziato, Lucio | |
| S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids. | 1.1 Articolo in rivista | 2001 | Alves, L. C.; Melo, R. L.; Sanderson, S. J.; Mottram, J. C.; Coombs, G. H.; Caliendo, Giuseppe; Santagada, V.; Juliano, L.; Juliano, M. A. | |
| Protease activated receptor-2 modulates myocardial ischemia reperfusion injury in the rat heart. | 1.1 Articolo in rivista | 2000 | Napoli, C; Cicala, Carla; Wallace, J; DE NIGRIS, F; Santagada, V; Caliendo, G; Franconi, F; Ignarro, L; Cirino, Giuseppe | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei | 1.1 Articolo in rivista | 2000 | Balboni, G.; Salvadori, S.; Guerrini, R.; Bianchi, C.; Santagada, V.; Caliendo, Giuseppe; Bryant, S. D.; Lazarus, L. H. | |
| 5-amino-2-hydroxybenzoic acid 4-(5-thioxo-5H-[1,2]dithiol-3yl)-phenyl ester (ATB-429), a hydrogen sulfide-releasing derivative of mesalamine, exerts antinociceptive effects in a model of postinflammatory hypersensitivity | 1.1 Articolo in rivista | 2006 | Distrutti, E; Sediari, L; Mencarelli, A; Renga, B; Orlandi, S; Russo, G; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, G; Wallace, Jl; Fiorucci, S. | |
| Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A. | |
| le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa |