SANTAGADA, VINCENZO
SANTAGADA, VINCENZO
DIPARTIMENTO DI FARMACIA
Foye's Principi di Chimica Farmaceutica
2014 R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
Anti-inflammatory peptides: an update and future perspectives
2002 Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M.
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators
1999 Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study.
1994 Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr.
1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Ialenti, Armando; Maffia, Pasquale; Albrizio, Stefania; Santini, Antonello
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning
2002 C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; G., Caliendo; M., Condorelli; Santagada, Vincenzo; Cirino, Giuseppe
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs.
2007 D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
Sequence and structure-activity relationship of a scorpion venom toxin with nitrergic activity in rabbit corpus cavernosum
2003 Teixeira, C. E.; Ifa, D. R.; Corso, G.; Santagada, V.; Caliendo, Giuseppe; Antunes, E.; DE NUCCI, G.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues
2000 Santagada, V.; Balboni, G.; Caliendo, Giuseppe; Guerrini, R.; Salvadori, S.; Bianchi, C.; Bryant, S. D.; Lazarus, L. H.
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation
2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC).
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents.
2011 Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.
2009 Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S.
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration.
2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Foye's Principi di Chimica Farmaceutica | 3.8 Traduzione di libro | 2014 | R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo | |
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa | |
Anti-inflammatory peptides: an update and future perspectives | 2.1 Contributo in volume (Capitolo o Saggio) | 2002 | Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M. | |
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators | 1.5 Abstract in rivista | 1999 | Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R | |
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. | 1.1 Articolo in rivista | 1994 | Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo | |
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Ialenti, Armando; Maffia, Pasquale; Albrizio, Stefania; Santini, Antonello | |
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning | 1.1 Articolo in rivista | 2002 | C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; G., Caliendo; M., Condorelli; Santagada, Vincenzo; Cirino, Giuseppe | |
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. | 1.1 Articolo in rivista | 2007 | D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA | |
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
Sequence and structure-activity relationship of a scorpion venom toxin with nitrergic activity in rabbit corpus cavernosum | 1.1 Articolo in rivista | 2003 | Teixeira, C. E.; Ifa, D. R.; Corso, G.; Santagada, V.; Caliendo, Giuseppe; Antunes, E.; DE NUCCI, G. | |
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G. | |
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues | 1.1 Articolo in rivista | 2000 | Santagada, V.; Balboni, G.; Caliendo, Giuseppe; Guerrini, R.; Salvadori, S.; Bianchi, C.; Bryant, S. D.; Lazarus, L. H. | |
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation | 1.1 Articolo in rivista | 2004 | Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe | |
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe | |
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. | 1.1 Articolo in rivista | 2011 | Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe | |
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. | 1.1 Articolo in rivista | 2009 | Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S. | |
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. | 1.1 Articolo in rivista | 2006 | Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G. |