COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis.
1994 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G.
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies
2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Synthesis and biological evaluation on human glioblastoma cells of novel pyrazolo[3,4-d]pyrimidine adenosine A(3) receptor antagonists
2010 Mugnaini, L.; La Motta, C.; Taliani, S; Simorini, F.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
The Boulton–Katritzky Reaction: A Kinetic Study of the Effect of 5-Nitrogen Substituents on the Rearrangement of Some (Z)-Phenylhydrazones of 3-Benzoyl-1,2,4-oxadiazoles
2014 Vincenzo, Frenna; Antonio Palumbo, Piccionello; Cosimelli, Barbara; Franco, Ghelfi; Domenico, Spinelli
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study.
2006 Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D.
Cardiovascular characterization of [1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-one-derivatives: selective myocardial calcium channel modulators.
2002 Budriesi, R; Cosimelli, Barbara; Ioan, P; Lanza, C. Z.; Spinelli, D; Chiarini, A.
Studies on Azole-to-Azole Interconversion. An Interesting Case of Absence of “Primary Steric Effect” in the Ring-degenerate Equilibration between ortho-Substituted 3-Aroylamino-5-methyl-1,2,4-oxadiazoles and 3-Acetylamino-5-aryl-1,2,4-oxadiazoles in Methanol.
2002 Buscemi, S; Frenna, V; Pace, A; Vivona, N; Cosimelli, Barbara; Spinelli, D.
Complete 1H (600 MHz) and 13C NMR Spectral Assignment of 3,4-bis[(3,4-Dimethoxyphenyl)methyl]dihydro-(3R-trans)-2(3H)-furanone (Matairesinol Dimethyl Ether), a Naturally Occurring Dibenzylbutyrolactone Lignan.
1993 Chimichi, S; Cosimelli, Barbara; BAMBAGIOTTI ALBERTI, M; Coran, S. A.; Vincieri, F. F.
From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety
2011 Cosimelli, Barbara
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents.
1999 Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G.
2-Phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one derivatives as a new class of adenosine receptor antagonists
2005 Primofiore, G.; Da Settimo, F.; Taliani, S.; Sergianni, V.; Simorini, F.; La Motta, C.; Marini, A. M.; Tuscano, D.; Martini, C.; Greco, Giovanni; Cosimelli, Barbara; Novellino, Ettore
Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation
2010 Taliani, S.; La Motta, C.; Mugnaini, L.; Simorini, F.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Cosimelli, Barbara; Greco, Giovanni; Limongelli, Vittorio; Marinelli, Luciana; Novellino, Ettore; Ciampi, O.; Daniele, S.; Trincavelli, M. L.; Martini, C.
Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands.
2007 Primofiore, G.; Taliani, S.; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Patrizi, M. P.; Sergianni, V.; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Calderone, V.; Montali, M.; Besnard, F.; Martini, C.
ABCB1 Structural Models, Molecular Docking, and Synthesis of New Oxadiazolothiazin-3-one Inhibitors
2013 C., Rosano; M., Viale; Cosimelli, Barbara; E., Severi; R., Gangemi; A., Ciogli; D., De Totero; D., Spinelli
Determination of the Absolute Configuration of a Chiral Oxadiazol-3-one Calcium Channel Blocker, Resolved by Using Chiral Chromatography, via Concerted Density Functional Theory Calculations of Its Vibrational Circular Dichroism, Electronic Circular Dichroism, and Optical Rotation.
2007 Stephens, P. J.; Devlin, F. J.; Gasparrini, F; Ciogli, A; Spinelli, D; Cosimelli, Barbara
A New Class of Selective Myocardial Calcium Channel Modulators. 2. The Role of the Acetal Chain in Oxadiazol-3-one Derivatives
2005 Budriesi, R; Carosati, E; Chiarini, A; Cosimelli, Barbara; Cruciani, G; Ioan, P; Spinelli, D; Spisani, R.
Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues
2004 Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S.
Diltiazem Analogues: The Last Ten Years on Structure Activity Relationships.
2007 Budriesi, R; Cosimelli, Barbara; Ioan, P; Carosati, E; Ugenti, M. P.; Spisani, R.
The First Kinetic Evidence for Acid Catalysis in a Monocyclic Rearrangement of Heterocycles: Conversion of the Z-Phenylhydrazone of 5-Amino-3-benzoyl-1,2,4-oxadiazole into N,5-Diphenyl-2H-1,2,3-triazol-4-ylurea
2002 Cosimelli, Barbara; Frenna, V; Guernelli, S; Lanza, C. Z.; Macaluso, G; Petrillo, G; Spinelli, D.
Mononuclear Heterocyclic Rearrangements. Part 16. Kinetic Study of the Rearrangement of Some ortho-Substituted Z-Phenylhydrazones of 3-Benzoyl-5-phenyl-1,2,4-oxadiazole into 2-Aryl-4-benzoylamino-5-phenyl-1,2,3-triazoles in Dioxane-Water and in Benzene.
1999 Frenna, V; Macaluso, G; Consiglio, G; Cosimelli, Barbara; Spinelli, D.