COSIMELLI, BARBARA

COSIMELLI, BARBARA  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 94 (tempo di esecuzione: 0.042 secondi).
Titolo Tipologia Data di pubblicazione Autore(i) File
Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies. 1.1 Articolo in rivista 2002 Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B.
A novel approach to the evaluation of the importance of steric and electronic effects in SNAr reactions: a computational, thermodynamic, 1H and 13C NMR study of “Meisenheimer-type” adducts in the benzo[b]thiophene series 1.1 Articolo in rivista 2010 Consiglio, G.; Cosimelli, Barbara; Guernelli, S.; Lanza, C. Z.; Sancassan, F.; Spinelli, D.; Stenta, M.
A New Convenient Route to 2-Oxoethoxycoumarins: Key Intermediates in the Synthesis of Natural Products. 1.1 Articolo in rivista 2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara
Unambiguous Structure Determination of Some Pyrazolo[1,5-a]pyrimidine Derivatives by Multinuclear NMR Spectroscopy. 1.1 Articolo in rivista 1992 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S.
On the reaction of 3-bromo-2-nitrobenzo[b]thiophene with some ortho-substituted anilines: an analysis of the products of reaction and of their NMR and MS properties 1.1 Articolo in rivista 2003 Cosimelli, Barbara; Lamartina, L; Lanza, C. Z.; Spinelli, D; Spisani, R; Vegna, F.
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists 4.3 Poster 2012 Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study. 1.1 Articolo in rivista 2006 Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D.
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy. 1.1 Articolo in rivista 1993 Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A.
Calcium Channel Antagonists Discovered by a Multidisciplinary Approach. 1.1 Articolo in rivista 2006 Carosati, E; Cruciani, G; Chiarini, A; Budriesi, R; Ioan, P; Spisani, R; Spinelli, D; Cosimelli, Barbara; Fusi, F; Frosini, M; Matucci, R; Gasparrini, F; Ciogli, A; Stephens, P. J.; Devlin, F. J.
New 5-(2-ethenylsubstituted)-3(2H)-furanones with in vitro antiproliferative activity 1.1 Articolo in rivista 2003 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Dallacqua, F.
Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers. 1.1 Articolo in rivista 1992 Chimichi, S; Cosimelli, Barbara
Ring-ring interconversion: the rearrangement of 6-(4-chlorophenyl)-3-methyl-5-nitrosoimidazo[2,1-b][1,3]thiazole into 8-(4-chlorophenyl)-8-hydroxy-5-methyl-8H-[1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-one. Elucidation of the reaction product through spectroscopic and X-ray crystal structure analysis. 1.1 Articolo in rivista 1997 Andreani, A; Billi, R; Cosimelli, Barbara; Mugnoli, A; Rambaldi, M; Spinelli, D.
Ring opening of 2-substituted 4-nitrothiophenes with pyrrolidine. Access to new functionalized nitro-unsaturated building blocks. 1.1 Articolo in rivista 2001 Dell'Erba, C; Gabellini, A; Novi, M; Petrillo, G; Tavani, C; Cosimelli, Barbara; Spinelli, D.
Diltiazem Analogues: The Last Ten Years on Structure Activity Relationships. 1.1 Articolo in rivista 2007 Budriesi, R; Cosimelli, Barbara; Ioan, P; Carosati, E; Ugenti, M. P.; Spisani, R.
Studies on Azole-to-Azole Interconversion. An Interesting Case of Absence of “Primary Steric Effect” in the Ring-degenerate Equilibration between ortho-Substituted 3-Aroylamino-5-methyl-1,2,4-oxadiazoles and 3-Acetylamino-5-aryl-1,2,4-oxadiazoles in Methanol. 1.1 Articolo in rivista 2002 Buscemi, S; Frenna, V; Pace, A; Vivona, N; Cosimelli, Barbara; Spinelli, D.
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies 8.02 Comunicazioni a Convegni o Seminari 2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Complete 1H (600 MHz) and 13C NMR Spectral Assignment of 3,4-bis[(3,4-Dimethoxyphenyl)methyl]dihydro-(3R-trans)-2(3H)-furanone (Matairesinol Dimethyl Ether), a Naturally Occurring Dibenzylbutyrolactone Lignan. 1.1 Articolo in rivista 1993 Chimichi, S; Cosimelli, Barbara; BAMBAGIOTTI ALBERTI, M; Coran, S. A.; Vincieri, F. F.
A New Class of Selective Myocardial Calcium Channel Modulators. 2. The Role of the Acetal Chain in Oxadiazol-3-one Derivatives 1.1 Articolo in rivista 2005 Budriesi, R; Carosati, E; Chiarini, A; Cosimelli, Barbara; Cruciani, G; Ioan, P; Spinelli, D; Spisani, R.
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation. 1.1 Articolo in rivista 2007 Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C.
First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate 1.1 Articolo in rivista 2008 Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A.