COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole.
1989 Chimichi, S; Cosimelli, Barbara
Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects
2012 Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E.
A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies.
1996 Cosimelli, Barbara; Neri, D; Roncucci, G.
New geiparvarin analogues from 7-(2-oxoethoxy)coumarins as efficient in vitro antitumoral agents.
2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Vedaldi, D; Dall'Acqua, F.
Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators
2014 Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini
Novel Irreversible Fluorescent Probes Targeting the 18kDa Translocator Protein: Synthesis and Biological Characterization.
2010 Taliani, S.; Da Pozzo, E.; Bellandi, M.; Bendinelli, S.; Pugliesi, I.; Simorini, F.; La Motta, C.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Martini, C.
On the reactivity of nitrosoimidazoles with acids (the Cusmano-Ruccia reaction): a continuous source of new ring-into-ring interconversion
2014 Cosimelli, Barbara; Vincenzo, Frenna; Mirella, Rambaldi; Elda, Severi; Domenico, Spinelli
Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives
2011 Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan
Playing with Opening and Closing of Heterocycles: Using the Cusmano-Ruccia Reaction to Develop a Novel Class of Oxadiazolothiazinones, Active as Calcium Channel Modulators and P-Glycoprotein Inhibitors
2014 Domenico, Spinelli; Roberta, Budriesi; Cosimelli, Barbara; Elda, Severi; Matteo, Micucci; Massimo, Baroni; Fabio, Fusi; Pierfranco, Ioan; Simon, Cross; Maria, Frosini; Simona, Saponara; Rosanna, Matucci; Camillo, Rosano; Maurizio, Viale; Alberto, Chiarini; Emanuele, Carosati
From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety
2011 Cosimelli, Barbara
Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines.
2003 Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D.
Cardiovascular characterization of [1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-one-derivatives: selective myocardial calcium channel modulators.
2002 Budriesi, R; Cosimelli, Barbara; Ioan, P; Lanza, C. Z.; Spinelli, D; Chiarini, A.
ABCB1 Structural Models, Molecular Docking, and Synthesis of New Oxadiazolothiazin-3-one Inhibitors
2013 C., Rosano; M., Viale; Cosimelli, Barbara; E., Severi; R., Gangemi; A., Ciogli; D., De Totero; D., Spinelli
Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues
2004 Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S.
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study.
2006 Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D.
New results on the reactivity of 5,6-diamino-4-hydroxy-2-mercaptopyrimidine
2004 Cosimelli, Barbara; Iadanza, M; Spisani, R; Novellino, Ettore
Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies.
2002 Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B.
New 5-(2-ethenylsubstituted)-3(2H)-furanones with in vitro antiproliferative activity
2003 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Dallacqua, F.
Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates
2009 Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D.
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole. | 1.1 Articolo in rivista | 1989 | Chimichi, S; Cosimelli, Barbara | |
| Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects | 1.1 Articolo in rivista | 2012 | Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E. | |
| A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies. | 1.1 Articolo in rivista | 1996 | Cosimelli, Barbara; Neri, D; Roncucci, G. | |
| New geiparvarin analogues from 7-(2-oxoethoxy)coumarins as efficient in vitro antitumoral agents. | 1.1 Articolo in rivista | 2002 | Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Vedaldi, D; Dall'Acqua, F. | |
| Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators | 1.1 Articolo in rivista | 2014 | Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini | |
| Novel Irreversible Fluorescent Probes Targeting the 18kDa Translocator Protein: Synthesis and Biological Characterization. | 1.1 Articolo in rivista | 2010 | Taliani, S.; Da Pozzo, E.; Bellandi, M.; Bendinelli, S.; Pugliesi, I.; Simorini, F.; La Motta, C.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Martini, C. | |
| On the reactivity of nitrosoimidazoles with acids (the Cusmano-Ruccia reaction): a continuous source of new ring-into-ring interconversion | 1.1 Articolo in rivista | 2014 | Cosimelli, Barbara; Vincenzo, Frenna; Mirella, Rambaldi; Elda, Severi; Domenico, Spinelli | |
| Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan | |
| Playing with Opening and Closing of Heterocycles: Using the Cusmano-Ruccia Reaction to Develop a Novel Class of Oxadiazolothiazinones, Active as Calcium Channel Modulators and P-Glycoprotein Inhibitors | 1.1 Articolo in rivista | 2014 | Domenico, Spinelli; Roberta, Budriesi; Cosimelli, Barbara; Elda, Severi; Matteo, Micucci; Massimo, Baroni; Fabio, Fusi; Pierfranco, Ioan; Simon, Cross; Maria, Frosini; Simona, Saponara; Rosanna, Matucci; Camillo, Rosano; Maurizio, Viale; Alberto, Chiarini; Emanuele, Carosati | |
| From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety | 8.02 Comunicazioni a Convegni o Seminari | 2011 | Cosimelli, Barbara | |
| Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines. | 1.1 Articolo in rivista | 2003 | Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D. | |
| Cardiovascular characterization of [1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-one-derivatives: selective myocardial calcium channel modulators. | 1.1 Articolo in rivista | 2002 | Budriesi, R; Cosimelli, Barbara; Ioan, P; Lanza, C. Z.; Spinelli, D; Chiarini, A. | |
| ABCB1 Structural Models, Molecular Docking, and Synthesis of New Oxadiazolothiazin-3-one Inhibitors | 1.1 Articolo in rivista | 2013 | C., Rosano; M., Viale; Cosimelli, Barbara; E., Severi; R., Gangemi; A., Ciogli; D., De Totero; D., Spinelli | |
| Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues | 1.1 Articolo in rivista | 2004 | Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S. | |
| Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study. | 1.1 Articolo in rivista | 2006 | Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D. | |
| New results on the reactivity of 5,6-diamino-4-hydroxy-2-mercaptopyrimidine | 1.1 Articolo in rivista | 2004 | Cosimelli, Barbara; Iadanza, M; Spisani, R; Novellino, Ettore | |
| Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies. | 1.1 Articolo in rivista | 2002 | Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B. | |
| New 5-(2-ethenylsubstituted)-3(2H)-furanones with in vitro antiproliferative activity | 1.1 Articolo in rivista | 2003 | Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Dallacqua, F. | |
| Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates | 1.1 Articolo in rivista | 2009 | Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D. | |
| L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. |