COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
1H and 13C NMR Study of the Pyrazolo[1,5-a]pyrimidine System.
1992 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S.
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis.
1994 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G.
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents.
1999 Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G.
A novel approach to the evaluation of the importance of steric and electronic effects in SNAr reactions: a computational, thermodynamic, 1H and 13C NMR study of “Meisenheimer-type” adducts in the benzo[b]thiophene series
2010 Consiglio, G.; Cosimelli, Barbara; Guernelli, S.; Lanza, C. Z.; Sancassan, F.; Spinelli, D.; Stenta, M.
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility
2011 Cosimelli, Barbara; S., Taliani; Greco, Giovanni; Novellino, Ettore; A., Sala; E., Severi; F., Da Settimo; C., La Motta; I., Pugliesi; L., Antonioli; M., Fornai; R., Colucci; C., Blandizzi; S., Daniele; M. L., Trincavelli; C., Martini
Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A1 adenosine receptor antagonists
2002 Novellino, E.; ABIGNENTE DI FRASSELLO, Enrico; Cosimelli, B.; Greco, Giovanni; Iadanza, M.; Laneri, S.; Lavecchia, A.; Rimoli, M. G.; DA SETTIMO, F.; Primofiore, G.; Tuscano, D.; Martini, C.
High Affinity Central Benzodiazepine Receptor Ligands: Synthesis and Biological Evaluation of a Series of Phenyltriazolobenzotriazindione Derivatives (PTBTs)
2005 Primofiore, G; DA SETTIMO, F; Taliani, S; Salerno, S; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Besnard, F; Costa, C; Montali, M; Martini, C.
Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine: A New Heterocyclic Ring System.
1990 Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
The First Kinetic Evidence for Acid Catalysis in a Monocyclic Rearrangement of Heterocycles: Conversion of the Z-Phenylhydrazone of 5-Amino-3-benzoyl-1,2,4-oxadiazole into N,5-Diphenyl-2H-1,2,3-triazol-4-ylurea
2002 Cosimelli, Barbara; Frenna, V; Guernelli, S; Lanza, C. Z.; Macaluso, G; Petrillo, G; Spinelli, D.
Ring-ring Interconversions of Nitrosoimidazoles. The Effect of Some Condensed Six-membered Rings on the Reactivity.
2000 Billi, R; Cosimelli, Barbara; Spinelli, D; Andreani, A; Leoni, A.
On the reaction of 3-bromo-2-nitrobenzo[b]thiophene with some ortho-substituted anilines: an analysis of the products of reaction and of their NMR and MS properties
2003 Cosimelli, Barbara; Lamartina, L; Lanza, C. Z.; Spinelli, D; Spisani, R; Vegna, F.
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation.
2007 Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C.
New geiparvarin analogues from 7-(2-oxoethoxy)coumarins as efficient in vitro antitumoral agents.
2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Vedaldi, D; Dall'Acqua, F.
Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines.
2003 Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D.
Carbon-13 NMR Studies on Azolopyridines. 3-The Isothiazolopyridine Systems.
1994 Chimichi, S; Cosimelli, Barbara; Tedeschi, P; Ponticelli, F.
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study.
2006 Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D.
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
Identification of anxiolytic/non sedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the GABAA alfa2 benzodiazepine receptor
2009 Taliani, S.; Cosimelli, Barbara; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Salerno, S.; Novellino, Ettore; Greco, Giovanni; Cosconati, S.; Marinelli, Luciana; Salvetti, F.; L’Abbate, G.; Trasciatti, S.; Montali, M.; Costa, B.; Martini, C.
Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands.
2007 Primofiore, G.; Taliani, S.; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Patrizi, M. P.; Sergianni, V.; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Calderone, V.; Montali, M.; Besnard, F.; Martini, C.
Mononuclear Heterocyclic Rearrangements. Part 16. Kinetic Study of the Rearrangement of Some ortho-Substituted Z-Phenylhydrazones of 3-Benzoyl-5-phenyl-1,2,4-oxadiazole into 2-Aryl-4-benzoylamino-5-phenyl-1,2,3-triazoles in Dioxane-Water and in Benzene.
1999 Frenna, V; Macaluso, G; Consiglio, G; Cosimelli, Barbara; Spinelli, D.
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
1H and 13C NMR Study of the Pyrazolo[1,5-a]pyrimidine System. | 1.1 Articolo in rivista | 1992 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S. | |
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis. | 1.1 Articolo in rivista | 1994 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G. | |
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents. | 6.1 Brevetto | 1999 | Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G. | |
A novel approach to the evaluation of the importance of steric and electronic effects in SNAr reactions: a computational, thermodynamic, 1H and 13C NMR study of “Meisenheimer-type” adducts in the benzo[b]thiophene series | 1.1 Articolo in rivista | 2010 | Consiglio, G.; Cosimelli, Barbara; Guernelli, S.; Lanza, C. Z.; Sancassan, F.; Spinelli, D.; Stenta, M. | |
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; S., Taliani; Greco, Giovanni; Novellino, Ettore; A., Sala; E., Severi; F., Da Settimo; C., La Motta; I., Pugliesi; L., Antonioli; M., Fornai; R., Colucci; C., Blandizzi; S., Daniele; M. L., Trincavelli; C., Martini | |
Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A1 adenosine receptor antagonists | 1.1 Articolo in rivista | 2002 | Novellino, E.; ABIGNENTE DI FRASSELLO, Enrico; Cosimelli, B.; Greco, Giovanni; Iadanza, M.; Laneri, S.; Lavecchia, A.; Rimoli, M. G.; DA SETTIMO, F.; Primofiore, G.; Tuscano, D.; Martini, C. | |
High Affinity Central Benzodiazepine Receptor Ligands: Synthesis and Biological Evaluation of a Series of Phenyltriazolobenzotriazindione Derivatives (PTBTs) | 1.1 Articolo in rivista | 2005 | Primofiore, G; DA SETTIMO, F; Taliani, S; Salerno, S; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Besnard, F; Costa, C; Montali, M; Martini, C. | |
Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine: A New Heterocyclic Ring System. | 1.1 Articolo in rivista | 1990 | Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S. | |
The First Kinetic Evidence for Acid Catalysis in a Monocyclic Rearrangement of Heterocycles: Conversion of the Z-Phenylhydrazone of 5-Amino-3-benzoyl-1,2,4-oxadiazole into N,5-Diphenyl-2H-1,2,3-triazol-4-ylurea | 1.1 Articolo in rivista | 2002 | Cosimelli, Barbara; Frenna, V; Guernelli, S; Lanza, C. Z.; Macaluso, G; Petrillo, G; Spinelli, D. | |
Ring-ring Interconversions of Nitrosoimidazoles. The Effect of Some Condensed Six-membered Rings on the Reactivity. | 1.1 Articolo in rivista | 2000 | Billi, R; Cosimelli, Barbara; Spinelli, D; Andreani, A; Leoni, A. | |
On the reaction of 3-bromo-2-nitrobenzo[b]thiophene with some ortho-substituted anilines: an analysis of the products of reaction and of their NMR and MS properties | 1.1 Articolo in rivista | 2003 | Cosimelli, Barbara; Lamartina, L; Lanza, C. Z.; Spinelli, D; Spisani, R; Vegna, F. | |
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation. | 1.1 Articolo in rivista | 2007 | Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C. | |
New geiparvarin analogues from 7-(2-oxoethoxy)coumarins as efficient in vitro antitumoral agents. | 1.1 Articolo in rivista | 2002 | Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Vedaldi, D; Dall'Acqua, F. | |
Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines. | 1.1 Articolo in rivista | 2003 | Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D. | |
Carbon-13 NMR Studies on Azolopyridines. 3-The Isothiazolopyridine Systems. | 1.1 Articolo in rivista | 1994 | Chimichi, S; Cosimelli, Barbara; Tedeschi, P; Ponticelli, F. | |
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study. | 1.1 Articolo in rivista | 2006 | Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D. | |
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. | |
Identification of anxiolytic/non sedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the GABAA alfa2 benzodiazepine receptor | 1.1 Articolo in rivista | 2009 | Taliani, S.; Cosimelli, Barbara; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Salerno, S.; Novellino, Ettore; Greco, Giovanni; Cosconati, S.; Marinelli, Luciana; Salvetti, F.; L’Abbate, G.; Trasciatti, S.; Montali, M.; Costa, B.; Martini, C. | |
Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands. | 1.1 Articolo in rivista | 2007 | Primofiore, G.; Taliani, S.; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Patrizi, M. P.; Sergianni, V.; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Calderone, V.; Montali, M.; Besnard, F.; Martini, C. | |
Mononuclear Heterocyclic Rearrangements. Part 16. Kinetic Study of the Rearrangement of Some ortho-Substituted Z-Phenylhydrazones of 3-Benzoyl-5-phenyl-1,2,4-oxadiazole into 2-Aryl-4-benzoylamino-5-phenyl-1,2,3-triazoles in Dioxane-Water and in Benzene. | 1.1 Articolo in rivista | 1999 | Frenna, V; Macaluso, G; Consiglio, G; Cosimelli, Barbara; Spinelli, D. |