PERISSUTTI, ELISA
PERISSUTTI, ELISA
DIPARTIMENTO DI FARMACIA
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands.
2002 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands.
2001 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study
1997 Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A.
Synthesis and Pharmacological Evaluation of a Set of N-[2-(Alkylamino)ethyl]benzotriazol-X-yl Isobutyramides Acting as Local Anesthetics.
1996 Caliendo, Giuseppe; Greco, Giovanni; MATTACE RASO, Giuseppina; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones.
2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Human Tissue Kallikrein S1 Subsite Recognition of Non-Natural Basic Amino Acids
2001 MELO ROBSON, L; POZZO ROSELI C., Barbosa; PIMENTA DANIEL, C; Perissutti, Elisa; Caliendo, Giuseppe; Santagada, Vincenzo; Juliano, Luiz; JULIANO MARIA, A.
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides.
1995 Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase
2000 Sautebin, L.; Rombol, L.; DI ROSA, M.; Caliendo, Giuseppe; Perissutti, Elisa; Grieco, G.; Severino, Beatrice; Santagada, Vincenzo
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
2006 Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G.
Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone
1992 Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R.
Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma
2005 B., Bicalho; G. C., Guzzo; S., Lilla; H. O., DOS SANTOS; G. D., Mendes; Caliendo, Giuseppe; Perissutti, Elisa; Aiello, Anna; Luciano, Paolo; Santagada, Vincenzo; A. S., Pereira; G., DE NUCCIA
Identification of a pepducin acting as S1P3 receptor antagonist
2013 Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Manganelli, Serena; Maggioni, Giada; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo | |
| Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo | |
| Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists | 1.1 Articolo in rivista | 2001 | Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa, | |
| The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
| Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A. | |
| Synthesis and Pharmacological Evaluation of a Set of N-[2-(Alkylamino)ethyl]benzotriazol-X-yl Isobutyramides Acting as Local Anesthetics. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; MATTACE RASO, Giuseppina; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo | |
| A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe | |
| Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe | |
| Human Tissue Kallikrein S1 Subsite Recognition of Non-Natural Basic Amino Acids | 1.1 Articolo in rivista | 2001 | MELO ROBSON, L; POZZO ROSELI C., Barbosa; PIMENTA DANIEL, C; Perissutti, Elisa; Caliendo, Giuseppe; Santagada, Vincenzo; Juliano, Luiz; JULIANO MARIA, A. | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
| Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo | |
| le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa | |
| Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase | 1.1 Articolo in rivista | 2000 | Sautebin, L.; Rombol, L.; DI ROSA, M.; Caliendo, Giuseppe; Perissutti, Elisa; Grieco, G.; Severino, Beatrice; Santagada, Vincenzo | |
| In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives | 1.1 Articolo in rivista | 2006 | Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G. | |
| Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone | 1.1 Articolo in rivista | 1992 | Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R. | |
| Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma | 1.1 Articolo in rivista | 2005 | B., Bicalho; G. C., Guzzo; S., Lilla; H. O., DOS SANTOS; G. D., Mendes; Caliendo, Giuseppe; Perissutti, Elisa; Aiello, Anna; Luciano, Paolo; Santagada, Vincenzo; A. S., Pereira; G., DE NUCCIA | |
| Identification of a pepducin acting as S1P3 receptor antagonist | 1.1 Articolo in rivista | 2013 | Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Manganelli, Serena; Maggioni, Giada; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa |