PERISSUTTI, ELISA
PERISSUTTI, ELISA
DIPARTIMENTO DI FARMACIA
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones.
2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6
2015 Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
Synthesis of benzamide derivatives and their evaluation as antiprion agents
2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
Synthesis and neurokinin antagonist activity of 2-benzylidene- and 2- benzyl-3-benzylamino quinuclidines
1993 Caliendo, Giuseppe; Greco, Giovanni; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Turbanti, L.; Renzetti, A. R.; Benedetti, E.; Pedone, C.; Santini, A.
Pharmacological characterization of benzotriazole derivatives active on the muscarinic receptor
1990 Meli, R.; Muccioli, G.; Perissutti, Elisa; Santagada, V.; Silipo, C.; Vittori, A.; Di, Carlo
Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives
1996 Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study
1997 Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A.
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators
1999 Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R
Synthesis and biological evaluation of proline derivatives as potential angiotensin converting enzyme inhibitor.
1996 G., Giugliano; Grieco, Paolo; Ialenti, Armando; M., Mottola; Perissutti, Elisa; Santagada, Vincenzo
Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone
1992 Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R.
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents.
2011 Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation
2012 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration.
2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe | |
| Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 | 1.1 Articolo in rivista | 2015 | Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano | |
| Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists | 1.1 Articolo in rivista | 2001 | Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa, | |
| Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
| Synthesis of benzamide derivatives and their evaluation as antiprion agents | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe | |
| Synthesis and neurokinin antagonist activity of 2-benzylidene- and 2- benzyl-3-benzylamino quinuclidines | 1.1 Articolo in rivista | 1993 | Caliendo, Giuseppe; Greco, Giovanni; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Turbanti, L.; Renzetti, A. R.; Benedetti, E.; Pedone, C.; Santini, A. | |
| Pharmacological characterization of benzotriazole derivatives active on the muscarinic receptor | 1.1 Articolo in rivista | 1990 | Meli, R.; Muccioli, G.; Perissutti, Elisa; Santagada, V.; Silipo, C.; Vittori, A.; Di, Carlo | |
| Molecular structures of quinuclidinic neurokinin antagonists: 2-(2-phenylbenzylidene)-3-(2-X-benzylamino) derivatives | 1.1 Articolo in rivista | 1996 | Santini, A; Benedetti, E.; Pedone, C.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Perissutti, Elisa | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A. | |
| le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa | |
| Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators | 1.5 Abstract in rivista | 1999 | Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R | |
| Synthesis and biological evaluation of proline derivatives as potential angiotensin converting enzyme inhibitor. | 1.1 Articolo in rivista | 1996 | G., Giugliano; Grieco, Paolo; Ialenti, Armando; M., Mottola; Perissutti, Elisa; Santagada, Vincenzo | |
| Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone | 1.1 Articolo in rivista | 1992 | Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R. | |
| Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. | 1.1 Articolo in rivista | 2011 | Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe | |
| The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
| New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe | |
| Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. | 1.1 Articolo in rivista | 2006 | Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G. |