PERISSUTTI, ELISA
PERISSUTTI, ELISA
DIPARTIMENTO DI FARMACIA
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer
2014 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Ciano, Antonio; Caliendo, Giuseppe; Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan.
1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands.
2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage.
2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs.
2007 D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
Racemic synthesis and solid phase peptide synthesis application of the chimeric Valine/Leucine derivative 2-amino-3,3,4-trimethyl-pentanoic acid
2014 M., Pelà; L., Del Zoppo; L., Allegri; E., Marzola; C., Trapella; C., Ruzza; G., Calo???; Perissutti, Elisa; Frecentese, Francesco; S., Salvadori; R., Guerrini
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators
1999 Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R
Synthesis and biological evaluation of proline derivatives as potential angiotensin converting enzyme inhibitor.
1996 G., Giugliano; Grieco, Paolo; Ialenti, Armando; M., Mottola; Perissutti, Elisa; Santagada, Vincenzo
Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study
1997 Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A.
Pharmacological characterization of benzotriazole derivatives active on the muscarinic receptor
1990 Meli, R.; Muccioli, G.; Perissutti, Elisa; Santagada, V.; Silipo, C.; Vittori, A.; Di, Carlo
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study.
1994 Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
2006 Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe | |
| 5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer | 1.1 Articolo in rivista | 2014 | Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Ciano, Antonio; Caliendo, Giuseppe; Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa | |
| Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania | |
| Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. | 1.1 Articolo in rivista | 2000 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R. | |
| Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G. | |
| Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G. | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. | 1.1 Articolo in rivista | 2007 | D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA | |
| Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists | 1.1 Articolo in rivista | 2001 | Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa, | |
| The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
| Racemic synthesis and solid phase peptide synthesis application of the chimeric Valine/Leucine derivative 2-amino-3,3,4-trimethyl-pentanoic acid | 1.1 Articolo in rivista | 2014 | M., Pelà; L., Del Zoppo; L., Allegri; E., Marzola; C., Trapella; C., Ruzza; G., Calo???; Perissutti, Elisa; Frecentese, Francesco; S., Salvadori; R., Guerrini | |
| Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators | 1.5 Abstract in rivista | 1999 | Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R | |
| Synthesis and biological evaluation of proline derivatives as potential angiotensin converting enzyme inhibitor. | 1.1 Articolo in rivista | 1996 | G., Giugliano; Grieco, Paolo; Ialenti, Armando; M., Mottola; Perissutti, Elisa; Santagada, Vincenzo | |
| Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A. | |
| Pharmacological characterization of benzotriazole derivatives active on the muscarinic receptor | 1.1 Articolo in rivista | 1990 | Meli, R.; Muccioli, G.; Perissutti, Elisa; Santagada, V.; Silipo, C.; Vittori, A.; Di, Carlo | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe | |
| Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. | 1.1 Articolo in rivista | 1994 | Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo | |
| Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
| In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives | 1.1 Articolo in rivista | 2006 | Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G. |