IRIS
CALIENDO, GIUSEPPE
 Distribuzione geografica
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Continente #
NA - Nord America 3.433
EU - Europa 2.704
AS - Asia 1.243
AF - Africa 73
SA - Sud America 15
Continente sconosciuto - Info sul continente non disponibili 4
Totale 7.472
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Nazione #
US - Stati Uniti d'America 3.380
IT - Italia 1.096
SG - Singapore 581
CN - Cina 410
DE - Germania 353
UA - Ucraina 267
FR - Francia 197
NL - Olanda 194
IE - Irlanda 181
FI - Finlandia 179
HK - Hong Kong 122
GB - Regno Unito 61
SE - Svezia 61
CI - Costa d'Avorio 53
CA - Canada 49
IN - India 44
RU - Federazione Russa 37
VN - Vietnam 29
JP - Giappone 19
TR - Turchia 19
MA - Marocco 16
ES - Italia 15
PL - Polonia 15
IR - Iran 13
BR - Brasile 11
BG - Bulgaria 10
AT - Austria 9
GR - Grecia 7
CH - Svizzera 4
EG - Egitto 4
EU - Europa 4
PT - Portogallo 4
SK - Slovacchia (Repubblica Slovacca) 4
CL - Cile 3
MX - Messico 3
BE - Belgio 2
SI - Slovenia 2
CZ - Repubblica Ceca 1
EE - Estonia 1
ID - Indonesia 1
JM - Giamaica 1
KR - Corea 1
LA - Repubblica Popolare Democratica del Laos 1
LT - Lituania 1
MK - Macedonia 1
MY - Malesia 1
NO - Norvegia 1
PH - Filippine 1
PK - Pakistan 1
RS - Serbia 1
VE - Venezuela 1
Totale 7.472
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Città #
Chandler 514
Singapore 491
Naples 306
Ashburn 296
Jacksonville 240
Santa Clara 234
Amsterdam 182
Millbury 162
Princeton 143
Hong Kong 122
Nanjing 110
Napoli 110
Woodbridge 104
Beijing 101
Menlo Park 76
Wilmington 69
Boston 63
Houston 61
Krefeld 57
Des Moines 47
Ottawa 43
Nanchang 35
Helsinki 30
Ann Arbor 29
Dong Ket 28
Bad Bellingen 25
Dearborn 23
Lawrence 23
Rome 22
Hebei 21
Milan 21
Norwalk 20
San Giorgio a Cremano 19
Jiaxing 18
Redwood City 18
Nuremberg 17
Seattle 17
Pozzuoli 16
Salerno 16
Tianjin 16
Casablanca 15
Dublin 14
Falkenstein 14
Indiana 14
Mugnano di Napoli 14
Shenyang 14
Falls Church 13
Augusta 12
Changsha 11
Trieste 11
Ardabil 10
Cambridge 10
Dallas 10
Cervino 9
Pune 9
Scunthorpe 9
Sofia 9
Boardman 8
Kronberg 8
Limerick 8
Roccarainola 8
San Mateo 8
Athens 7
Bari 7
Lappeenranta 7
Los Angeles 7
Mumbai 7
Orange 7
Pisa 7
Vienna 7
Zola Predosa 7
Caserta 6
Hangzhou 6
Jena 6
Krakow 6
Kunming 6
Rho 6
Warsaw 6
Bacoli 5
Bologna 5
Cicciano 5
Council Bluffs 5
Ercolano 5
Falcone 5
Formia 5
Moscow 5
Redmond 5
Toronto 5
Afragola 4
Bratislava 4
Casoria 4
Frankfurt am Main 4
Fucecchio 4
Guangzhou 4
Lanzhou 4
Mountain View 4
New York 4
Porto 4
Santiago De Compostela 4
Shanghai 4
Totale 4.386
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Nome #
7-nitro-5-fenil-1(pirrolidin-1-ilmetil)-1H-benzo[e][1,4] diazepin-2(3H)-one ed altri composti derivati delle benzodiazepine 320
1,2,4-Thiadiazolidin-3,5-diones as novel hydrogen sulfide donors 210
Foye's Principi di Chimica Farmaceutica 203
Design, Synthesis and Biological Evaluation of Novel N-Arylpiperazines Containing a 4,5-Dihydrothiazole Ring 185
MONTELUKAST ESTERS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 103
Chemical Composition of PM10 at Urban Sites in Naples (Italy) 87
Design of Sphingosine Kinases Inhibitors: Challenges and Recent Developments 84
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors 78
Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents 77
Antagonizing S1P3 receptor with cell-penetrating pepducins in skeletal muscle fibrosis 73
Activity of human kallikrein-related peptidase 6 (KLK6) on substrates containing sequences of basic amino acids. Is it a processing protease? 70
Synthesis of Arylpiperazine Derivatives as Protease Activated Receptor 1 Antagonists and Their Evaluation as Antiproliferative Agents 70
Heavy Metals Size Distribution in PM10 and Environmental-Sanitary Risk Analysis in Acerra (Italy) 70
The Role of 5-HT1A Receptor in the Cancer as a New Opportunity in Medicinal Chemistry 67
Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies 66
New 5-HT1A, 5HT2Aand 5HT2Creceptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation 63
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. 62
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. 62
7-nitro-5-phenyl-1-(pyrrolidin-1-ylmethyl)-1H-benzo[E][1,4]diazepin-2(3H)-one and other benzodiazepine derivatives 61
BUDESONIDE 21-PHOSPHATE SALTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 61
Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma 60
Synthesis, biological activity and conformational study of 1,4-benzoxazine dderivatives as potassium channel modulators. 60
Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis 59
Synthesis and in Vitro Screening of New Series of 2,6-Dipeptidyl-anthraquinones: Influence of Side Chain Length on HIV-1 Nucleocapsid Inhibitors 59
Identification of a novel selective CSE inhibitor through a combined pharmacological and metabolomic approach 59
Hybrids between H2S-donors and betamethasone 17-valerate or triamcinolone acetonide inhibit mast cell degranulation and promote hyperpolarization of bronchial smooth muscle cells 59
Pyrrolobenzoxazepinone (PBO) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further Structure-Activity Relationship Studies and Identification of More Potent Broad Spectrum HIV-1 RT Inhibitors with Antiviral Activity. 58
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic ligands containing an isonicotinic nucleus 57
Synthesis, Chiral Resolution and Enantiomers Absolute Configuration of 4-Nitropropranolol and 7-Nitropropranolol 56
A valuable synthesis of reduced peptide bond by microwave irradiation 56
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 56
Pharmacological characterization of the newly synthesized 5-amino-N-butyl-2-(4-ethoxyphenoxy)-benzamide hydrochloride (BED) as a potent NCX3 inhibitor that worsens anoxic injury in cortical neurons, organotypic hippocampal cultures, and ischemic brain 56
A suitable 1,2,4-oxadiazoles synthesis by microwave irradiation 55
Microwave Assisted Organic Synthesis of Heterocycles in Aqueous Media: Recent Advances in Medicinal Chemistry 55
Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation 54
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV 53
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 53
Non-Natural Linker Configuration in 2,6-Dipeptidyl-Anthraquinones Enhances the Inhibition of TAR RNA Binding/Annealing Activities by HIV-1 NC and Tat Proteins 53
Evidence for a protective role played by Na+-Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats 52
Identification of a pepducin acting as S1P3 receptor antagonist 51
Synthesis of Nα-Fmoc N,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC) 50
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 50
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. 50
Synthesis of 6-beta-D-glucosyl and 6-nitroxy (-)-galanthamine derivatives as acetylcholinesterase inhibitors 49
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 49
Propafenone quantification in human plasma by high-performance liquid chromatography coupled with electrospray tandem mass spectrometry in a bioequivalence study 49
74) Nevirapine quantification in human plasma by high-performance liquid chromatography coupled to electrospray tandem mass spectrometry. Application to bioequivalence study 48
Synthesis, docking studies, and pharmacological evaluation of 5HT 2C ligands containing the N′-cyanoisonicotinamidine or N′-cyanopicolinamidine nucleus 48
Montelukast salts and pharmaceutical compositions containing the same 48
Microwave Solvent Free Regioselective 1,3 Dipolar Cycloaddition in the Synthesis of 1,4 Substituted [1,2,3]-Triazoles as Amide Bond Isosteres 47
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. 47
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. 47
Design, synthesis and biological evaluation of TAR and cTAR binders as HIV-​1 nucleocapsid inhibitors 47
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues 46
The application of microwave irradiation as new convenient synthetic procedure in drug discovery 46
Fragment-based de novo design of a cystathionine γ-lyase selective inhibitor blocking hydrogen sulfide production 46
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. 45
Anti-inflammatory peptides: an update and future perspectives 45
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). 45
Peptidi e Peptidomimetici: Progettazione, sintesi e caratterizzazione, applicazioni di nuove strategie sintetiche (chimica combinatoriale, microonde) 45
Benzotriazole derivatives active on plant growth: Design, synthesis and physicochemical properties 45
Development validation of LC-MS/MS method and determination of pharmacokinetic parameters of the stroke neuroprotectant neurounina-1 in beagle dog plasma after intravenous administration 45
New Serotoninergic Ligands Containing Indolic and Methyl Indolic Nuclei: Synthesis and In Vitro Pharmacological Evaluation 45
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 44
New 5-Hydroxytryptamine1A Receptor Ligands Containing a Norbornene Nucleus: Synthesis and in Vitro Pharmacological Evaluation 43
Protease activated receptor-2 modulates myocardial ischemia reperfusion injury in the rat heart. 42
Synthesis of 2-Methyl-3-indolylacetic Derivatives as Anti-Inflammatory Agents That Inhibit Preferentially Cyclooxygenase 1 without Gastric Damage 42
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer 42
Synthesis and In Vitro Pharmacological Evaluation of Novel 2-Hydroxypropyl-4-arylpiperazine Derivatives as Serotoninergic Ligands 42
Budesonide 21-phosphate sodium salt for use as anti-inflammatory or anti-asthmatic agent. 41
Shape-dependent effects in a series of aromatic nitro compounds acting as mutagenic agents on S.typhimurium TA98. 41
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation 41
Synthesis and Biological Activity of Benzotriazole Derivatives Structurally Related to Trazodone. 41
A hydrogen sulfide-releasing dexamethasone derivative attenuates atopic dermatitis severity signs and the associated oxidative stress markers in mice 41
X-ray Structural Analysis of Ethyl [2,2-dimethyl-6-(D2-thiazolin-2-yl)-4H-1,4-benzoxazin-3-one-4-yl]butyrate. 40
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. 40
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation 40
Structure-activity relationships study of isothiocyanates for H2S releasing properties: 3-Pyridyl-isothiocyanate as a new promising cardioprotective agent 40
Beneficial Effects of Two Hydrogen Sulfide (H2S)-Releasing Derivatives of Dexamethasone with Antioxidant Activity on Atopic Dermatitis in Mice 39
Efficient Microwave Combinatorial Parallel and Non Parallel Synthesis of N-Alkylated Glycine Methyl Esters as Peptide Building Blocks 39
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. 39
Pharmacokinetic profile of atenolol aspirinate 39
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents 39
Biological data in sets of benzotriazole derivatives active as plant growth regulators 39
Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides. 38
Synthesis of benzamide derivatives and their evaluation as antiprion agents 38
HYBRIDS BETWEEN H2S-DONORS AND BETAMETHASONE 17-VALERATE OR TRIAMCINOLONE ACETONIDE: IN VITRO EFFECT IN ASTHMA TREATMENT 38
Synthesis, docking studies, and pharmacological evaluation of 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands 37
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase 36
Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands 36
Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids. 36
Design and synthesis of potential b-sheet nucleatorsvia Suzuki coupling reaction 36
Novel tools for the elucidation of physio-pathological role of H2S 36
PCB levels in adipose tissue of dogs from illegal dumping sites in Campania region (Italy) 36
Involvement of 3′,5′-cyclic inosine monophosphate in cystathionine γ-lyase-dependent regulation of the vascular tone 36
Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis 35
Neurounina-1, a Novel Compound that Increases Na+/Ca2+ Exchanger Activity, Effectively Protects Against Stroke Damage 35
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. 34
Synthesis and Antiinflammatory-Analgesic Profile of 1-Methyl-2-(4-X-benzoyl)imidazole-5-carboxylic Acids. 34
Na+/Ca2+ exchanger in Na+ efflux-Ca2+ influx mode of operation exerts a neuroprotective role in cellular models of in vitro anoxia and in vivo cerebral ischemia. 33
Totale 5.703
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Categoria #
all - tutte 33.840
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 33.840
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020303 0 0 0 0 0 0 29 13 14 78 74 95
2020/2021651 21 55 51 58 73 64 68 14 66 16 106 59
2021/20221.193 14 9 12 151 16 60 7 48 173 106 246 351
2022/20231.262 192 151 25 134 104 113 19 83 168 183 62 28
2023/20241.438 45 143 246 31 32 28 47 370 208 29 170 89
2024/20251.293 254 298 58 103 101 333 146 0 0 0 0 0
Totale 7.786