IRIS
CALIENDO, GIUSEPPE
 Distribuzione geografica
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Continente #
AS - Asia 7.121
NA - Nord America 6.486
EU - Europa 6.290
SA - Sud America 857
AF - Africa 211
OC - Oceania 7
Continente sconosciuto - Info sul continente non disponibili 6
Totale 20.978
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Nazione #
US - Stati Uniti d'America 6.246
SG - Singapore 3.190
RU - Federazione Russa 2.399
IT - Italia 1.413
CN - Cina 1.384
VN - Vietnam 1.299
BR - Brasile 681
DE - Germania 582
HK - Hong Kong 524
FR - Francia 432
UA - Ucraina 294
FI - Finlandia 249
NL - Olanda 244
IE - Irlanda 185
GB - Regno Unito 165
IN - India 143
CA - Canada 131
JP - Giappone 127
SE - Svezia 80
AR - Argentina 63
MX - Messico 63
BD - Bangladesh 56
CI - Costa d'Avorio 54
PL - Polonia 54
ZA - Sudafrica 53
ES - Italia 50
KR - Corea 44
IQ - Iraq 41
TR - Turchia 38
PH - Filippine 33
TH - Thailandia 31
GR - Grecia 30
PK - Pakistan 30
MA - Marocco 29
EC - Ecuador 28
ID - Indonesia 28
CO - Colombia 22
AT - Austria 21
VE - Venezuela 20
IR - Iran 18
LT - Lituania 18
TW - Taiwan 17
JO - Giordania 15
PY - Paraguay 14
UZ - Uzbekistan 14
BG - Bulgaria 13
TN - Tunisia 12
CL - Cile 11
EG - Egitto 11
SA - Arabia Saudita 11
UY - Uruguay 11
IL - Israele 10
AE - Emirati Arabi Uniti 7
BE - Belgio 7
JM - Giamaica 7
KE - Kenya 7
LB - Libano 7
MY - Malesia 7
PS - Palestinian Territory 7
SN - Senegal 7
CH - Svizzera 6
ET - Etiopia 6
KZ - Kazakistan 6
NI - Nicaragua 6
SY - Repubblica araba siriana 6
AU - Australia 5
AZ - Azerbaigian 5
DZ - Algeria 5
NP - Nepal 5
PT - Portogallo 5
TT - Trinidad e Tobago 5
AL - Albania 4
AM - Armenia 4
AO - Angola 4
BA - Bosnia-Erzegovina 4
BW - Botswana 4
CZ - Repubblica Ceca 4
EE - Estonia 4
EU - Europa 4
KG - Kirghizistan 4
PE - Perù 4
RS - Serbia 4
SK - Slovacchia (Repubblica Slovacca) 4
BS - Bahamas 3
CM - Camerun 3
DM - Dominica 3
HN - Honduras 3
HU - Ungheria 3
PR - Porto Rico 3
SI - Slovenia 3
BB - Barbados 2
BO - Bolivia 2
CR - Costa Rica 2
DO - Repubblica Dominicana 2
GA - Gabon 2
GE - Georgia 2
GN - Guinea 2
GT - Guatemala 2
HR - Croazia 2
KW - Kuwait 2
Totale 20.936
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Città #
Singapore 1.527
San Jose 1.021
Ashburn 630
Moscow 571
Chandler 514
Hong Kong 501
Naples 455
Beijing 451
Ho Chi Minh City 364
Hanoi 290
Santa Clara 268
Jacksonville 241
Amsterdam 202
The Dalles 186
Lauterbourg 169
Hefei 166
Millbury 162
Princeton 143
Los Angeles 135
Nanjing 111
Napoli 110
Woodbridge 104
Tokyo 98
Munich 94
São Paulo 81
Buffalo 80
Boston 79
Houston 76
Menlo Park 76
Redondo Beach 73
Wilmington 70
Council Bluffs 66
Dallas 66
New York 66
Frankfurt am Main 60
Krefeld 57
Haiphong 54
Da Nang 49
Des Moines 49
Helsinki 48
Ottawa 47
Turku 46
Milan 37
Nuremberg 37
Orem 37
Falkenstein 36
Nanchang 36
Rome 36
Warsaw 35
Brooklyn 34
Mexico City 33
Toronto 32
Ann Arbor 29
Chicago 28
Dong Ket 28
Seoul 27
Tianjin 27
Atlanta 26
Seattle 26
Bad Bellingen 25
London 25
Rio de Janeiro 25
Chennai 24
Dearborn 23
Johannesburg 23
Lawrence 23
Hebei 21
Hải Dương 21
Montreal 21
Thessaloniki 21
Casablanca 20
Norwalk 20
Stockholm 20
Biên Hòa 19
Can Tho 19
Phoenix 19
San Giorgio a Cremano 19
Dublin 18
Jiaxing 18
Redwood City 18
Salerno 18
San Francisco 18
Manchester 17
Mumbai 17
Pozzuoli 16
Baghdad 15
Shenyang 15
Changsha 14
Denver 14
Indiana 14
Mugnano di Napoli 14
Amman 13
Falls Church 13
Poplar 13
Augusta 12
Lahore 12
Lappeenranta 12
Vienna 12
Bangkok 11
Tashkent 11
Totale 10.923
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Nome #
7-nitro-5-fenil-1(pirrolidin-1-ilmetil)-1H-benzo[e][1,4] diazepin-2(3H)-one ed altri composti derivati delle benzodiazepine 391
1,2,4-Thiadiazolidin-3,5-diones as novel hydrogen sulfide donors 360
Foye's Principi di Chimica Farmaceutica 304
Design, Synthesis and Biological Evaluation of Novel N-Arylpiperazines Containing a 4,5-Dihydrothiazole Ring 299
Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents 192
Pharmacological characterization of the newly synthesized 5-amino-N-butyl-2-(4-ethoxyphenoxy)-benzamide hydrochloride (BED) as a potent NCX3 inhibitor that worsens anoxic injury in cortical neurons, organotypic hippocampal cultures, and ischemic brain 191
Chemical Composition of PM10 at Urban Sites in Naples (Italy) 182
Activity of human kallikrein-related peptidase 6 (KLK6) on substrates containing sequences of basic amino acids. Is it a processing protease? 179
MONTELUKAST ESTERS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 168
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors 167
Design of Sphingosine Kinases Inhibitors: Challenges and Recent Developments 167
Antagonizing S1P3 receptor with cell-penetrating pepducins in skeletal muscle fibrosis 165
Identification of a pepducin acting as S1P3 receptor antagonist 164
Heavy Metals Size Distribution in PM10 and Environmental-Sanitary Risk Analysis in Acerra (Italy) 161
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic ligands containing an isonicotinic nucleus 159
Synthesis and in Vitro Screening of New Series of 2,6-Dipeptidyl-anthraquinones: Influence of Side Chain Length on HIV-1 Nucleocapsid Inhibitors 156
Synthesis of Arylpiperazine Derivatives as Protease Activated Receptor 1 Antagonists and Their Evaluation as Antiproliferative Agents 153
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 152
New 5-HT1A, 5HT2Aand 5HT2Creceptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation 151
The Role of 5-HT1A Receptor in the Cancer as a New Opportunity in Medicinal Chemistry 151
Synthesis, docking studies, and pharmacological evaluation of 5HT 2C ligands containing the N′-cyanoisonicotinamidine or N′-cyanopicolinamidine nucleus 150
Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation 149
Synthesis, Chiral Resolution and Enantiomers Absolute Configuration of 4-Nitropropranolol and 7-Nitropropranolol 147
Non-Natural Linker Configuration in 2,6-Dipeptidyl-Anthraquinones Enhances the Inhibition of TAR RNA Binding/Annealing Activities by HIV-1 NC and Tat Proteins 147
A New Process for the Synthesis of Budesonide 21-Phosphate and Evaluation in a Murine Model of Inflammation 145
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 144
Development validation of LC-MS/MS method and determination of pharmacokinetic parameters of the stroke neuroprotectant neurounina-1 in beagle dog plasma after intravenous administration 142
Hybrids between H2S-donors and betamethasone 17-valerate or triamcinolone acetonide inhibit mast cell degranulation and promote hyperpolarization of bronchial smooth muscle cells 142
HYBRIDS BETWEEN H2S-DONORS AND BETAMETHASONE 17-VALERATE OR TRIAMCINOLONE ACETONIDE: IN VITRO EFFECT IN ASTHMA TREATMENT 142
Propafenone quantification in human plasma by high-performance liquid chromatography coupled with electrospray tandem mass spectrometry in a bioequivalence study 141
Isothiocyanate-Corticosteroid Conjugates against asthma: Unity makes strength 139
A new nano-encapsulated TSPO ligand reduces neuroinflammation and improves cognitive functions in Alzheimer's disease model 139
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer 138
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 137
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation 137
PCB levels in adipose tissue of dogs from illegal dumping sites in Campania region (Italy) 137
Synthesis and In Vitro Pharmacological Evaluation of Novel 2-Hydroxypropyl-4-arylpiperazine Derivatives as Serotoninergic Ligands 136
Microwave Assisted Organic Synthesis of Heterocycles in Aqueous Media: Recent Advances in Medicinal Chemistry 136
3-Nitroatenolol: First Synthesis, Chiral Resolution and Enantiomers’ Absolute Configuration 135
Design, synthesis and biological evaluation of TAR and cTAR binders as HIV-​1 nucleocapsid inhibitors 135
Synthesis, biological activity and conformational study of 1,4-benzoxazine dderivatives as potassium channel modulators. 134
Prednisone-hydrogen sulfide releasing hybrid shows improved therapeutic profile in asthma 133
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. 133
Evidence for a protective role played by Na+-Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats 133
Novel tools for the elucidation of physio-pathological role of H2S 132
Beneficial Effects of Two Hydrogen Sulfide (H2S)-Releasing Derivatives of Dexamethasone with Antioxidant Activity on Atopic Dermatitis in Mice 131
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. 131
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. 131
New Serotoninergic Ligands Containing Indolic and Methyl Indolic Nuclei: Synthesis and In Vitro Pharmacological Evaluation 131
Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies 130
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 129
Newly Synthesized Indolylacetic Derivatives Reduce Tumor Necrosis Factor-Mediated Neuroinflammation and Prolong Survival in Amyotrophic Lateral Sclerosis Mice 129
Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma 128
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 128
7-nitro-5-phenyl-1-(pyrrolidin-1-ylmethyl)-1H-benzo[E][1,4]diazepin-2(3H)-one and other benzodiazepine derivatives 128
Synthesis, Docking Studies and Pharmacological Evaluation of Serotoninergic Ligands Containing a 5-Norbornene-2-Carboxamide Nucleus 127
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. 126
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. 126
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV 125
Synthesis of benzamide derivatives and their evaluation as antiprion agents 125
Pyrrolobenzoxazepinone (PBO) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further Structure-Activity Relationship Studies and Identification of More Potent Broad Spectrum HIV-1 RT Inhibitors with Antiviral Activity. 124
Involvement of 3′,5′-cyclic inosine monophosphate in cystathionine γ-lyase-dependent regulation of the vascular tone 124
Budesonide 21-phosphate sodium salt for use as anti-inflammatory or anti-asthmatic agent. 123
Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis 123
Synthesis and Biological Activity of Benzotriazole Derivatives Structurally Related to Trazodone. 123
Anti-inflammatory peptides: an update and future perspectives 121
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). 121
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. 121
H2s donors and their use in medicinal chemistry 121
BUDESONIDE 21-PHOSPHATE SALTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 120
Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides. 119
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators 119
Fragment-based de novo design of a cystathionine γ-lyase selective inhibitor blocking hydrogen sulfide production 116
Structure-activity relationships study of isothiocyanates for H2S releasing properties: 3-Pyridyl-isothiocyanate as a new promising cardioprotective agent 116
Design, Synthesis and Evaluation of Novel Molecular Hybrids between Antiglaucoma Drugs and H2S Donors 115
Arylpiperazine Derivatives and Cancer: A New Challenge in Medicinal Chemistry 114
A valuable synthesis of reduced peptide bond by microwave irradiation 114
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. 113
Identification of a novel selective CSE inhibitor through a combined pharmacological and metabolomic approach 113
Trends in h2s-donors chemistry and their effects in cardiovascular diseases 113
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica 112
Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids. 111
Kallikrein Protease Activated Receptor (PAR) Axis: An Attractive Target for Drug Development 111
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents 111
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. 110
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. 110
Synthesis and Antiinflammatory-Analgesic Profile of 1-Methyl-2-(4-X-benzoyl)imidazole-5-carboxylic Acids. 110
Synthesis of Nα-Fmoc N,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC) 109
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. 109
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. 109
Synthesis, docking studies, and pharmacological evaluation of 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands 109
Peptidi e Peptidomimetici: Progettazione, sintesi e caratterizzazione, applicazioni di nuove strategie sintetiche (chimica combinatoriale, microonde) 108
74) Nevirapine quantification in human plasma by high-performance liquid chromatography coupled to electrospray tandem mass spectrometry. Application to bioequivalence study 107
Serotoninergic receptor ligands improve Tamoxifen effectiveness on breast cancer cells 107
Microwave Solvent Free Regioselective 1,3 Dipolar Cycloaddition in the Synthesis of 1,4 Substituted [1,2,3]-Triazoles as Amide Bond Isosteres 106
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase 106
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. 106
H2S donating corticosteroids: Design, synthesis and biological evaluation in a murine model of asthma 106
New 5-Hydroxytryptamine1A Receptor Ligands Containing a Norbornene Nucleus: Synthesis and in Vitro Pharmacological Evaluation 105
The application of microwave irradiation as new convenient synthetic procedure in drug discovery 105
Totale 13.960
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Categoria #
all - tutte 65.520
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 65.520
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021181 0 0 0 0 0 0 0 0 0 16 106 59
2021/20221.193 14 9 12 151 16 60 7 48 173 106 246 351
2022/20231.262 192 151 25 134 104 113 19 83 168 183 62 28
2023/20241.438 45 143 246 31 32 28 47 370 208 29 170 89
2024/20255.360 254 298 58 103 101 333 501 362 363 609 1.922 456
2025/20269.459 1.072 678 1.112 904 1.670 380 1.148 534 1.349 612 0 0
Totale 21.312