CALIENDO, GIUSEPPE
 Distribuzione geografica
Continente #
AS - Asia 7.281
NA - Nord America 7.136
EU - Europa 6.444
SA - Sud America 879
Continente sconosciuto - Info sul continente non disponibili 343
AF - Africa 215
OC - Oceania 7
Totale 22.305
Nazione #
US - Stati Uniti d'America 6.840
SG - Singapore 3.206
RU - Federazione Russa 2.399
IT - Italia 1.544
CN - Cina 1.429
VN - Vietnam 1.305
BR - Brasile 692
DE - Germania 584
HK - Hong Kong 528
FR - Francia 434
UA - Ucraina 294
FI - Finlandia 249
NL - Olanda 248
IE - Irlanda 185
GB - Regno Unito 170
CA - Canada 165
IN - India 144
BD - Bangladesh 132
JP - Giappone 128
SE - Svezia 80
MX - Messico 67
AR - Argentina 65
PL - Polonia 55
CI - Costa d'Avorio 54
ES - Italia 53
ZA - Sudafrica 53
KR - Corea 46
IQ - Iraq 41
TR - Turchia 38
PH - Filippine 33
TH - Thailandia 32
EC - Ecuador 31
GR - Grecia 31
ID - Indonesia 30
PK - Pakistan 30
MA - Marocco 29
CO - Colombia 25
VE - Venezuela 22
AT - Austria 21
IR - Iran 18
LT - Lituania 18
TW - Taiwan 17
JO - Giordania 15
PY - Paraguay 14
UZ - Uzbekistan 14
BG - Bulgaria 13
JM - Giamaica 12
TN - Tunisia 12
UY - Uruguay 12
CL - Cile 11
EG - Egitto 11
IL - Israele 11
SA - Arabia Saudita 11
MY - Malesia 10
AE - Emirati Arabi Uniti 8
NI - Nicaragua 8
BE - Belgio 7
CH - Svizzera 7
KE - Kenya 7
LB - Libano 7
PS - Palestinian Territory 7
SN - Senegal 7
AL - Albania 6
DZ - Algeria 6
ET - Etiopia 6
KZ - Kazakistan 6
NP - Nepal 6
SY - Repubblica araba siriana 6
TT - Trinidad e Tobago 6
AU - Australia 5
AZ - Azerbaigian 5
CR - Costa Rica 5
CZ - Repubblica Ceca 5
PT - Portogallo 5
SK - Slovacchia (Repubblica Slovacca) 5
AM - Armenia 4
AO - Angola 4
BA - Bosnia-Erzegovina 4
BW - Botswana 4
EE - Estonia 4
EU - Europa 4
HN - Honduras 4
KG - Kirghizistan 4
PE - Perù 4
PR - Porto Rico 4
RS - Serbia 4
SV - El Salvador 4
BS - Bahamas 3
BZ - Belize 3
CM - Camerun 3
DM - Dominica 3
GT - Guatemala 3
HU - Ungheria 3
SC - Seychelles 3
SI - Slovenia 3
BB - Barbados 2
BO - Bolivia 2
DO - Repubblica Dominicana 2
GA - Gabon 2
GE - Georgia 2
Totale 21.923
Città #
Singapore 1.539
San Jose 1.111
Ashburn 675
Moscow 571
Chandler 516
Hong Kong 504
Naples 495
Beijing 468
Ho Chi Minh City 365
Santa Clara 300
Hanoi 293
Jacksonville 243
Amsterdam 202
The Dalles 186
Lauterbourg 169
Hefei 166
Millbury 162
Los Angeles 152
Princeton 143
Nanjing 111
Napoli 110
Woodbridge 105
Tokyo 98
Munich 94
Council Bluffs 88
Buffalo 87
New York 86
São Paulo 84
Houston 83
Dallas 82
Boston 80
Menlo Park 76
Redondo Beach 73
Wilmington 71
Frankfurt am Main 60
Krefeld 57
Haiphong 54
Milan 51
Da Nang 50
Des Moines 49
Helsinki 48
Ottawa 48
Turku 46
Rome 44
Brooklyn 40
Orem 38
Nuremberg 37
Toronto 37
Falkenstein 36
Mexico City 36
Nanchang 36
Warsaw 35
Chicago 32
Ann Arbor 29
Atlanta 29
Dong Ket 28
Seattle 28
London 27
Seoul 27
Tianjin 27
Bad Bellingen 25
Montreal 25
Rio de Janeiro 25
Chennai 24
Dearborn 23
Johannesburg 23
Lawrence 23
Phoenix 23
Norwalk 22
Hebei 21
Hải Dương 21
Thessaloniki 21
Casablanca 20
Stockholm 20
Biên Hòa 19
Can Tho 19
Manchester 19
Salerno 19
San Francisco 19
San Giorgio a Cremano 19
Dublin 18
Jiaxing 18
Mumbai 18
Redwood City 18
Pozzuoli 16
Baghdad 15
Denver 15
Shenyang 15
Changsha 14
Indiana 14
Mugnano di Napoli 14
Amman 13
Falls Church 13
Poplar 13
Augusta 12
Bangkok 12
Lahore 12
Lappeenranta 12
Vienna 12
Guangzhou 11
Totale 11.332
Nome #
7-nitro-5-fenil-1(pirrolidin-1-ilmetil)-1H-benzo[e][1,4] diazepin-2(3H)-one ed altri composti derivati delle benzodiazepine 393
1,2,4-Thiadiazolidin-3,5-diones as novel hydrogen sulfide donors 364
Foye's Principi di Chimica Farmaceutica 309
Design, Synthesis and Biological Evaluation of Novel N-Arylpiperazines Containing a 4,5-Dihydrothiazole Ring 302
Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents 213
Activity of human kallikrein-related peptidase 6 (KLK6) on substrates containing sequences of basic amino acids. Is it a processing protease? 209
A new nano-encapsulated TSPO ligand reduces neuroinflammation and improves cognitive functions in Alzheimer's disease model 202
Pharmacological characterization of the newly synthesized 5-amino-N-butyl-2-(4-ethoxyphenoxy)-benzamide hydrochloride (BED) as a potent NCX3 inhibitor that worsens anoxic injury in cortical neurons, organotypic hippocampal cultures, and ischemic brain 197
Chemical Composition of PM10 at Urban Sites in Naples (Italy) 192
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors 182
Design of Sphingosine Kinases Inhibitors: Challenges and Recent Developments 173
MONTELUKAST ESTERS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 173
Identification of a pepducin acting as S1P3 receptor antagonist 171
Antagonizing S1P3 receptor with cell-penetrating pepducins in skeletal muscle fibrosis 169
HYBRIDS BETWEEN H2S-DONORS AND BETAMETHASONE 17-VALERATE OR TRIAMCINOLONE ACETONIDE: IN VITRO EFFECT IN ASTHMA TREATMENT 168
Heavy Metals Size Distribution in PM10 and Environmental-Sanitary Risk Analysis in Acerra (Italy) 164
The Role of 5-HT1A Receptor in the Cancer as a New Opportunity in Medicinal Chemistry 163
A New Process for the Synthesis of Budesonide 21-Phosphate and Evaluation in a Murine Model of Inflammation 161
Synthesis and in Vitro Screening of New Series of 2,6-Dipeptidyl-anthraquinones: Influence of Side Chain Length on HIV-1 Nucleocapsid Inhibitors 160
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic ligands containing an isonicotinic nucleus 160
Synthesis, docking studies, and pharmacological evaluation of 5HT 2C ligands containing the N′-cyanoisonicotinamidine or N′-cyanopicolinamidine nucleus 156
Synthesis, Chiral Resolution and Enantiomers Absolute Configuration of 4-Nitropropranolol and 7-Nitropropranolol 154
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 154
New 5-HT1A, 5HT2Aand 5HT2Creceptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation 154
Synthesis of Arylpiperazine Derivatives as Protease Activated Receptor 1 Antagonists and Their Evaluation as Antiproliferative Agents 153
Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation 152
Isothiocyanate-Corticosteroid Conjugates against asthma: Unity makes strength 151
Propafenone quantification in human plasma by high-performance liquid chromatography coupled with electrospray tandem mass spectrometry in a bioequivalence study 149
Non-Natural Linker Configuration in 2,6-Dipeptidyl-Anthraquinones Enhances the Inhibition of TAR RNA Binding/Annealing Activities by HIV-1 NC and Tat Proteins 149
Development validation of LC-MS/MS method and determination of pharmacokinetic parameters of the stroke neuroprotectant neurounina-1 in beagle dog plasma after intravenous administration 147
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 145
Hybrids between H2S-donors and betamethasone 17-valerate or triamcinolone acetonide inhibit mast cell degranulation and promote hyperpolarization of bronchial smooth muscle cells 145
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer 144
PCB levels in adipose tissue of dogs from illegal dumping sites in Campania region (Italy) 144
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation 143
Prednisone-hydrogen sulfide releasing hybrid shows improved therapeutic profile in asthma 142
Design, synthesis and biological evaluation of TAR and cTAR binders as HIV-​1 nucleocapsid inhibitors 141
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 140
3-Nitroatenolol: First Synthesis, Chiral Resolution and Enantiomers’ Absolute Configuration 138
Microwave Assisted Organic Synthesis of Heterocycles in Aqueous Media: Recent Advances in Medicinal Chemistry 138
Newly Synthesized Indolylacetic Derivatives Reduce Tumor Necrosis Factor-Mediated Neuroinflammation and Prolong Survival in Amyotrophic Lateral Sclerosis Mice 138
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. 137
Evidence for a protective role played by Na+-Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats 137
Synthesis and In Vitro Pharmacological Evaluation of Novel 2-Hydroxypropyl-4-arylpiperazine Derivatives as Serotoninergic Ligands 137
Novel tools for the elucidation of physio-pathological role of H2S 136
New Serotoninergic Ligands Containing Indolic and Methyl Indolic Nuclei: Synthesis and In Vitro Pharmacological Evaluation 136
Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma 135
7-nitro-5-phenyl-1-(pyrrolidin-1-ylmethyl)-1H-benzo[E][1,4]diazepin-2(3H)-one and other benzodiazepine derivatives 135
Beneficial Effects of Two Hydrogen Sulfide (H2S)-Releasing Derivatives of Dexamethasone with Antioxidant Activity on Atopic Dermatitis in Mice 134
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 134
Synthesis, biological activity and conformational study of 1,4-benzoxazine dderivatives as potassium channel modulators. 134
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. 134
Arylpiperazine Derivatives and Cancer: A New Challenge in Medicinal Chemistry 133
Synthesis, Docking Studies and Pharmacological Evaluation of Serotoninergic Ligands Containing a 5-Norbornene-2-Carboxamide Nucleus 133
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. 133
Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies 132
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 130
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. 129
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV 129
Involvement of 3′,5′-cyclic inosine monophosphate in cystathionine γ-lyase-dependent regulation of the vascular tone 129
Design, Synthesis and Evaluation of Novel Molecular Hybrids between Antiglaucoma Drugs and H2S Donors 128
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. 128
Synthesis of benzamide derivatives and their evaluation as antiprion agents 128
Synthesis and Biological Activity of Benzotriazole Derivatives Structurally Related to Trazodone. 127
Budesonide 21-phosphate sodium salt for use as anti-inflammatory or anti-asthmatic agent. 126
H2s donors and their use in medicinal chemistry 126
Pyrrolobenzoxazepinone (PBO) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further Structure-Activity Relationship Studies and Identification of More Potent Broad Spectrum HIV-1 RT Inhibitors with Antiviral Activity. 125
Development and evaluation of nanostructured systems for cutaneous delivery of H2S-releasing corticosteroids for skin inflammatory diseases 124
Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis 124
Anti-inflammatory peptides: an update and future perspectives 124
BUDESONIDE 21-PHOSPHATE SALTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 124
Trends in h2s-donors chemistry and their effects in cardiovascular diseases 124
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica 123
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). 122
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. 122
Structure-activity relationships study of isothiocyanates for H2S releasing properties: 3-Pyridyl-isothiocyanate as a new promising cardioprotective agent 122
Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides. 121
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators 121
Fragment-based de novo design of a cystathionine γ-lyase selective inhibitor blocking hydrogen sulfide production 119
A valuable synthesis of reduced peptide bond by microwave irradiation 118
Synthesis of Nα-Fmoc N,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC) 116
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. 116
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents 116
Identification of a novel selective CSE inhibitor through a combined pharmacological and metabolomic approach 116
The identification of adenylyl cyclase modulators as potential receptors for 6-nitrodopamine in human-induced pluripotent stem cell (hiPSC)-derived cardiomyocytes and their relevance in heart inotropism 115
Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids. 114
Serotoninergic receptor ligands improve Tamoxifen effectiveness on breast cancer cells 114
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. 113
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. 112
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. 112
Kallikrein Protease Activated Receptor (PAR) Axis: An Attractive Target for Drug Development 112
Synthesis, docking studies, and pharmacological evaluation of 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands 112
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. 111
Synthesis and Antiinflammatory-Analgesic Profile of 1-Methyl-2-(4-X-benzoyl)imidazole-5-carboxylic Acids. 111
New 5-Hydroxytryptamine1A Receptor Ligands Containing a Norbornene Nucleus: Synthesis and in Vitro Pharmacological Evaluation 110
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues 110
Peptidi e Peptidomimetici: Progettazione, sintesi e caratterizzazione, applicazioni di nuove strategie sintetiche (chimica combinatoriale, microonde) 110
Enhanced efficacy of formoterol-montelukast salt in relieving asthma features and in preserving β2-agonists rescue therapy 109
Microwave Solvent Free Regioselective 1,3 Dipolar Cycloaddition in the Synthesis of 1,4 Substituted [1,2,3]-Triazoles as Amide Bond Isosteres 109
H2S donating corticosteroids: Design, synthesis and biological evaluation in a murine model of asthma 109
Totale 14.562
Categoria #
all - tutte 74.370
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 74.370


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/20221.179 0 9 12 151 16 60 7 48 173 106 246 351
2022/20231.262 192 151 25 134 104 113 19 83 168 183 62 28
2023/20241.438 45 143 246 31 32 28 47 370 208 29 170 89
2024/20255.360 254 298 58 103 101 333 501 362 363 609 1.922 456
2025/202610.099 1.072 678 1.112 904 1.670 380 1.148 534 1.349 680 324 248
2026/2027353 223 130 0 0 0 0 0 0 0 0 0 0
Totale 22.305